BGT1-IN-9 is the first small-molecule substrate identified with high selectivity for BGT1 over the three other GAT subtypes. It also acts as a M1 muscarinic agonist. References: Al-Khawaja A, Haugaard AS, Marek A, Loffler R, Thiesen L, Santiveri M, Damgaard M, Bundgaard C, Frolund B, Wellendorph P. Pharmacological Characterization of [(3)H]ATPCA as a Substrate for Studying the Functional Role of the Betaine/GABA Transporter 1 and the Creatine Transporter. ACS Chem Neurosci. 2018 Mar 21;9(3):545-554. doi: 10.1021/acschemneuro.7b00351. Epub 2017 Nov 22. PubMed PMID: 29131576.

纯度：≥98%

CAS：185444-92-2