生物活性
ENOblock (AP-III-a4)是一种新颖的小分子，是第一个直接结合烯醇酶并抑制其活性的非底物类似物（IC50 = 0.576 uM）；在体内抑制癌细胞的转移。
化学数据
| 目录号 | A11840 |
| M. Wt | 594.72 |
| Formula | C31H43FN8O3 |
| Purity | >99% |
| Storage | Store lyophilized at -20ºC, keep desiccated.
In lyophilized form, the chemical is stable for36 months.
In solution, store at -20ºC and use within3 monthsto prevent loss of potency. Aliquot to avoid multiple freeze/thaw cycles. |
| CAS No. | 1177827-73-4 |
| SMILES | C1CCC(CC1)CNC2=NC(=NC(=N2)NCC3=CC=C(C=C3)F)NC4=CC=C(C=C4)CC(=O)NCCOCCOCCN |
储备液配制
| Concentration / Solvent Volume / Mass | 1 mg | 5 mg | 10 mg |
| 0.1 mM | 16.81 mL | 84.07 mL | 168.15 mL |
| 0.5 mM | 3.36 mL | 16.81 mL | 33.63 mL |
| 1 mM | 1.68 mL | 8.41 mL | 16.81 mL |
| 5 mM | 0.34 mL | 1.68 mL | 3.36 mL |
*The above data is based on the productmolecular weight 594.72. Batch specific molecular weights may vary from batch to batch due to solvent of hydration, which will affect the solvent volumes required to prepare stock solutions.
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