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Azilsartan(TAK-536)
本产品不向个人销售,仅用作科学研究,不用于任何人体实验及非科研性质的动物实验。
Azilsartan(TAK-536)图片
CAS NO:147403-03-0
包装与价格:
包装价格(元)
10mg电议
25mg电议
50mg电议
100mg电议
10mM * 1mL in DMSO电议

产品名称
TAK536
产品介绍

生物活性

Azilsartan (TAK-536)是一种用于治疗高血压的血管紧张素II受体拮抗剂。

靶点信息

AT1 receptor
2.6 nM

化学数据

目录号A11775
作用机制Blocker (阻断剂)
M. Wt456.5
FormulaC25H20N4O5
Purity>99%
Storage

Store lyophilized at -20ºC, keep desiccated.
In lyophilized form, the chemical is stable for36 months.
In solution, store at -20ºC and use within3 monthsto prevent loss of potency. Aliquot to avoid multiple freeze/thaw cycles.

CAS No.147403-03-0
SynonymsTAK536
SMILESCCOC1=NC2=CC=CC(=C2N1CC3=CC=C(C=C3)C4=CC=CC=C4C5=NC(=O)ON5)C(=O)O

溶解度

In vitro (25°C)DMSO78 mg/mL (170.88 mM)
WaterInsoluble
EthanolInsoluble
In vivo30% PEG400+0.5% Tween80+5% propylene glycol28 mg/mL
*<1 mg/ml means slightly soluble or insoluble.
*Please note that Adooq tests the solubility of all compounds in-house, and the actual solubility may differ slightly from published values. This is normal and is due to slight batch-to-batch variations.

储备液配制

Concentration / Solvent Volume / Mass1 mg5 mg10 mg
0.1 mM21.91 mL109.53 mL219.06 mL
0.5 mM4.38 mL21.91 mL43.81 mL
1 mM2.19 mL10.95 mL21.91 mL
5 mM0.44 mL2.19 mL4.38 mL

*The above data is based on the productmolecular weight 456.5 . Batch specific molecular weights may vary from batch to batch due to solvent of hydration, which will affect the solvent volumes required to prepare stock solutions.