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Laropiprant(MK0524)
本产品不向个人销售,仅用作科学研究,不用于任何人体实验及非科研性质的动物实验。
Laropiprant(MK0524)图片
CAS NO:571170-77-9
包装与价格:
包装价格(元)
5mg电议
10mg电议
25mg电议
50mg电议

产品名称
Cardaptive, MK 0524, MK-0524
产品介绍

生物活性

Laropiprant (MK0524)与烟酸合用可降低血液胆固醇。是一种有效的,选择性的 DP receptor 拮抗剂,Ki 值为 0.57 nM,对 TP 受体的 Ki 值为 2.95 nM。

化学数据

目录号A11483
作用机制Inhibitor (抑制剂)
M. Wt435.9
FormulaC21H19ClFNO4S
Purity>99%
Storage

Store lyophilized at -20ºC, keep desiccated.
In lyophilized form, the chemical is stable for36 months.
In solution, store at -20ºC and use within3 monthsto prevent loss of potency. Aliquot to avoid multiple freeze/thaw cycles.

CAS No.571170-77-9
SynonymsCardaptive, MK 0524, MK-0524
SMILESCS(=O)(=O)C1=C2C(=CC(=C1)F)C3=C(N2CC4=CC=C(C=C4)Cl)[C@H](CC3)CC(=O)O

储备液配制

Concentration / Solvent Volume / Mass1 mg5 mg10 mg
0.1 mM22.94 mL114.71 mL229.41 mL
0.5 mM4.59 mL22.94 mL45.88 mL
1 mM2.29 mL11.47 mL22.94 mL
5 mM0.46 mL2.29 mL4.59 mL

*The above data is based on the productmolecular weight 435.9 . Batch specific molecular weights may vary from batch to batch due to solvent of hydration, which will affect the solvent volumes required to prepare stock solutions.