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Istradefylline(KW-6002)
本产品不向个人销售,仅用作科学研究,不用于任何人体实验及非科研性质的动物实验。
Istradefylline(KW-6002)图片
CAS NO:155270-99-8
包装与价格:
包装价格(元)
5mg电议
10mg电议
25mg电议
50mg电议

产品名称
KW-6002,KW6002
产品介绍

生物活性

Istradefylline (KW-6002)是A2A受体的选择性拮抗剂。

靶点信息

Adenosine A2A receptor
2.2 nM(Ki)

化学数据

目录号A11451
作用机制Antagonist (拮抗剂)
M. Wt384.4
FormulaC20H24N4O4
Purity>99%
Storage

Store lyophilized at -20ºC, keep desiccated.
In lyophilized form, the chemical is stable for36 months.
In solution, store at -20ºC and use within3 monthsto prevent loss of potency. Aliquot to avoid multiple freeze/thaw cycles.

CAS No.155270-99-8
SynonymsKW-6002,KW6002
SMILESCCN1C2=C(C(=O)N(C1=O)CC)N(C(=N2)/C=C/C3=CC(=C(C=C3)OC)OC)C

溶解度

In vitro (25°C)DMSO5 mg/mL (13 mM)
WaterInsoluble
EthanolInsoluble
In vivo30% propylene glycol, 5% Tween 80, 65% D5W28 mg/mL
*<1 mg/ml means slightly soluble or insoluble.
*Please note that Adooq tests the solubility of all compounds in-house, and the actual solubility may differ slightly from published values. This is normal and is due to slight batch-to-batch variations.

储备液配制

Concentration / Solvent Volume / Mass1 mg5 mg10 mg
0.1 mM26.01 mL130.07 mL260.15 mL
0.5 mM5.2 mL26.01 mL52.03 mL
1 mM2.6 mL13.01 mL26.01 mL
5 mM0.52 mL2.6 mL5.2 mL

*The above data is based on the productmolecular weight 384.4 . Batch specific molecular weights may vary from batch to batch due to solvent of hydration, which will affect the solvent volumes required to prepare stock solutions.