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GSK 525762A(I-BET-762)
本产品不向个人销售,仅用作科学研究,不用于任何人体实验及非科研性质的动物实验。
GSK 525762A(I-BET-762)图片
CAS NO:1260907-17-2
包装与价格:
包装价格(元)
5mg电议
10mg电议
25mg电议
50mg电议
10mM * 1mL in DMSO电议

产品名称
GSK-525762A, GSK525762A
产品介绍

生物活性

GSK 525762A (I-BET-762)是BET(溴域和末端外)家族的小分子抑制剂。

靶点信息

BET proteins (Cell-free assay)
35 nM

化学数据

目录号A11440
作用机制Inhibitor (抑制剂)
M. Wt423.9
FormulaC22H22ClN5O2
Purity>99%
Storage

Store lyophilized at -20ºC, keep desiccated.
In lyophilized form, the chemical is stable for36 months.
In solution, store at -20ºC and use within3 monthsto prevent loss of potency. Aliquot to avoid multiple freeze/thaw cycles.

CAS No.1260907-17-2
SynonymsGSK-525762A, GSK525762A
SMILESCCNC(=O)C[C@H]1C2=NN=C(N2C3=C(C=C(C=C3)OC)C(=N1)C4=CC=C(C=C4)Cl)C

溶解度

In vitroDMSO72 mg/mL (169.84 mM)
WaterInsoluble
EthanolWarmed: 36 mg/mL (84.92 mM)
*<1 mg/ml means slightly soluble or insoluble.
*Please note that Adooq tests the solubility of all compounds in-house, and the actual solubility may differ slightly from published values. This is normal and is due to slight batch-to-batch variations.

储备液配制

Concentration / Solvent Volume / Mass1 mg5 mg10 mg
0.1 mM23.59 mL117.95 mL235.9 mL
0.5 mM4.72 mL23.59 mL47.18 mL
1 mM2.36 mL11.8 mL23.59 mL
5 mM0.47 mL2.36 mL4.72 mL

*The above data is based on the productmolecular weight 423.9. Batch specific molecular weights may vary from batch to batch due to solvent of hydration, which will affect the solvent volumes required to prepare stock solutions.