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Flumazenil
本产品不向个人销售,仅用作科学研究,不用于任何人体实验及非科研性质的动物实验。
Flumazenil图片
CAS NO:78755-81-4
包装与价格:
包装价格(元)
50mg电议
100mg电议
200mg电议
500mg电议

产品名称
Ro 15-1788
产品介绍

生物活性

Flumazenil是竞争性抑制GABA/苯二氮卓受体复合物上苯二氮卓识别位点的活性。Flumazenil在一些活性动物模型中是弱部分激动剂,但在人类中很少或没有激动剂活性。

靶点信息

GABAA receptor

化学数据

目录号A10397
作用机制Antagonist (拮抗剂)
M. Wt303.3
FormulaC15H14FN3O3
Purity>99%
Storage

Store lyophilized at -20ºC, keep desiccated.
In lyophilized form, the chemical is stable for36 months.
In solution, store at -20ºC and use within3 monthsto prevent loss of potency. Aliquot to avoid multiple freeze/thaw cycles.

CAS No.78755-81-4
SynonymsRo 15-1788
SMILESCCOC(=O)c1ncn2c1CN(C)C(=O)c1c2ccc(c1)F

溶解度

In vitroDMSO4 mg/mL (13.18 mM)
WaterInsoluble
EthanolInsoluble
*<1 mg/ml means slightly soluble or insoluble.
*Please note that Adooq tests the solubility of all compounds in-house, and the actual solubility may differ slightly from published values. This is normal and is due to slight batch-to-batch variations.

储备液配制

Concentration / Solvent Volume / Mass1 mg5 mg10 mg
0.1 mM32.97 mL164.85 mL329.71 mL
0.5 mM6.59 mL32.97 mL65.94 mL
1 mM3.3 mL16.49 mL32.97 mL
5 mM0.66 mL3.3 mL6.59 mL

*The above data is based on the productmolecular weight 303.3 . Batch specific molecular weights may vary from batch to batch due to solvent of hydration, which will affect the solvent volumes required to prepare stock solutions.