CGP 35348 is a selective, brain penetrant GABAB receptor antagonist (IC50 = 34 μM as measured in rat cortical membranes). CGP 35348 has a higher affinity for postsynaptic versus presynaptic receptors. References: Gillani Q, Ali M, Iqbal F. Effect of GABA(B) receptor antagonists (CGP 35348 and CGP 55845) on serum interleukin 6 and 18 concentrations in albino mice following neonatal hypoxia ischemia insult. Pak J Pharm Sci. 2016 Sep;29(5):1503-1508. PubMed PMID: 27731803.

纯度：≥98%

CAS：123690-79-9