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Psora-4
本产品不向个人销售,仅用作科学研究,不用于任何人体实验及非科研性质的动物实验。
Psora-4图片
CAS NO:724709-68-6
规格:≥98%
包装与价格:
包装价格(元)
5mg电议
10mg电议
25mg电议

产品介绍
Psora-4 is a novel, potent and selective small-molecule inhibitor of voltage-gated potassium channels - Kv1.3 with EC50 of 3 nM. It binds preferentially to the C-type inactivated state of the channel, similar to the activity of CP 339818, and displays 17- to 70-fold selectivity over closely-related KV1 channels (KV1, KV2, KV4 and KV7); exhibits activity at KV1.5 (IC50 = 7.7 nM). Suppresses proliferation of human and rat myelin-specific effector memory T cells (EC50 values are 25 and 60 nM respectively).