GSK9311 HCl, a less active analog of GSK6853, can be used as a negative control. GSK9311 HCl inhibits BRPF bromodomain with pIC50 values of 6.0 and 4.3 for BRPF1 and BRPF2, respectively. References: [1]. Bamborough P, et al. GSK6853, a Chemical Probe for Inhibition of the BRPF1 Bromodomain. ACS Med Chem Lett. 2016 May 9;7(6):552-7.

纯度：≥98%

CAS：2253733-09-2