High affinity and potent ghrelin receptor inverse agonist (Ki values are 4.9 and 31 nM in COS7 and HEK293T cells, respectively). Blocks ghrelin receptor-mediated Gq- and G13-dependent signaling pathways.

1394288-22-2

C51H67N9O6

902.13

K-(D-1-Nal)-FwLL-NH2

H2O:2 mg/mL
Powder: -20°C for 3 years
In solvent: -80°C for 2 years