3-Bromocytisine 是一种有效的 nAChR 激动剂,对 hα4β4、hα4β2 和 hα7 的 IC50值分别为0.28、0.30 和 31.6 nM。
产品描述
3-Bromocytisine is an effective agonist of nAChR (IC50s: 0.28, 0.30 and 31.6 nM for hα4β4, hα4β2, and hα7).
体外活性
3-Bromocytisine shows different effects on high and low ACh sensitivity α4β2 nAChRs with EC50s are 8 and 50 nM, respectively [2].
Cas No.
207390-14-5
分子式
C11H13BrN2O
分子量
269.14
别名
3-Br-cytisine;(-)-3-Bromocytisine;(-)-9-Bromocytisine;3-Bromocytisine
储存和溶解度
(< 1 mg/ml refers to the product slightly soluble or insoluble )
Powder: -20°C for 3 years
In solvent: -80°C for 2 years