MMP-2/MMP-9-IN-1 是一种高选择性、口服有效的 IV 型胶原酶 (MMP-9和MMP-2) 抑制剂，对 MMP-9 和 MMP-2 的IC50分别为 0.24 和 0.3 1μM。MMP-2/MMP-9-IN-1 在肿瘤生长和转移的动物模型中具有口服活性，可用于癌症研究。

MMP-2/MMP-9-IN-1 is a highly selective, orally active and potent type IV collagenase ( MMP-9 and MMP-2 ) inhibitor with IC 50 s of 0.24 and 0.31 μM for MMP-9 and MMP-2, respectively. In addition, MMP-2/MMP-9-IN-1 is orally active in animal models of tumor growth and metastasis which has the potential for the treatment of cancer [1].

193807-58-8

C21H19NO4S

381.44

MMP-2/MMP-9 Inhibitor I

(< 1 mg/ml refers to the product slightly soluble or insoluble )
Powder: -20°C for 3 years
In solvent: -80°C for 2 years