GPR40 agonist 5 (化合物 I-14) 是一种口服有效的GPR40(G 蛋白偶联受体 40) 激动剂,其EC50值为 47 nM。GPR40 agonist 5 可降低血糖水平,改善糖耐量。GPR40 agonist 5 对 2 型糖尿病小鼠的高血糖状态有充足的控制作用。
产品描述
GPR40 agonist 5 (compound I-14) is an orally active and potent GPR40 (G protein coupled receptor 40) agonist, with an EC 50 of 47 nM. GPR40 agonist 5 decreases the levels of blood glucose and improves the glucose tolerance. GPR40 agonist 5 has sufficient effectiveness for the control of hyperglycemia state in type 2 diabetic mice [1].
Cas No.
2443384-60-7
分子式
C27H24N2O4
分子量
440.49
储存和溶解度
(< 1 mg/ml refers to the product slightly soluble or insoluble )
Powder: -20°C for 3 years
In solvent: -80°C for 2 years