Raloxifene 6-Monomethyl Ether (Compound 7) is a Raloxifene derivative that inhibits estrogen receptor α . Raloxifene 4-Monomethyl Ether inhibits MCF-7 cells with an IC 50 of 250 nM and a pIC 50 of 6.6.

Raloxifene 6-Monomethyl Ether (Compound 7) is a Raloxifene derivative with a methoxy group on C6. Raloxifene 6-Monomethyl Ether holds poor ICsub>50 value because of disruption to the hydrogen bond network and steric disfavor[1].

178451-13-3

C29H29NO4S

487.61

Raloxifene 6-Monomethyl Ether

(< 1 mg/ml refers to the product slightly soluble or insoluble )
Powder: -20°C for 3 years
In solvent: -80°C for 2 years