PERK-IN-2 is a potent inhibitor of PERK(IC50 of 0.2 nM).

PERK-IN-2 inhibits PERK autophosphorylation(IC50 ranging from 0.03?0.1 μM ,in A459 cells )[1].

1337531-83-5

C23H18F3N5O

437.42

PERK-IN-2

(< 1 mg/ml refers to the product slightly soluble or insoluble )
Powder: -20°C for 3 years
In solvent: -80°C for 2 years