Mesdopetam hemitartrate 是一种多巴胺D3受体拮抗剂 (Ki=90 nM;IC50=9.8 μM),具有稳定精神运动的作用,可用于帕金森病的运动和精神并发症的研究。
产品描述
Mesdopetam hemitartrate is an antagonist of dopamine D3 receptor (Ki=90 nM; IC50=9.8 μM for human recombinant D3 receptor). It has psychomotor stabilizing properties.
Cas No.
2562346-14-7
分子式
C28H42F2N2O12S2
分子量
700.77
别名
IRL790 hemitartrate;1-Propanamine, N-[2-[3-fluoro-5-(methylsulfonyl)phenoxy]ethyl]-, (2R,3R)-2,3-dihydroxybutanedioate (2:1);Mesdopetam hemitartrate
储存和溶解度
DMSO:20 mg/mL (28.54 mM),Need ultrasonic
Powder: -20°C for 3 years
In solvent: -80°C for 2 years