Cystathionine-γ-lyase-IN-1 是一个选择性的胱硫醚-γ-裂解酶 (CSE) 抑制剂，其IC50 值为 6.3 μM。

Cystathionine-γ-lyase-IN-1 is a selective inhibitor of cystathionine γ-lyase (CSE) enzyme (IC50= 6.3 μM).

Cystathionine-γ-lyase-IN-1 (100 μM) completely abrogates L-cysteine-induced vasorelaxation. Cystathionine-γ-lyase-IN-1 (100 μM; 30 minutes) significantly inhibits the increased H2S production stimulated by L-cysteine in mouse aorta homogenates[1].

2165706-30-7

C7H8N2O2S

184.22

SHIP-2a;Cystathionine-γ-lyase-IN-1

DMSO:16.2 mg/mL (87.9 mM),Need ultrasonic and warming
Ethanol:8.1 mg/mL (44.0 mM),Need ultrasonic and warming
Powder: -20°C for 3 years
In solvent: -80°C for 2 years