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NS 383
本产品不向个人销售,仅用作科学研究,不用于任何人体实验及非科研性质的动物实验。
NS 383图片
CAS NO:309711-59-9
包装:5 mg
市场价:7000元

产品介绍

产品描述

ASIC blocker (IC50 values are 0.44, 2.1 μM and no effect at rat ASIC1a, ASIC3 and ASIC2a, respectively: IC50 value = 0.12 μM at human ASIC1a with no effect at ASIC2a or ASIC3). Inhibition was also observed at heteromeric ASIC channels (IC50 values are 0.79, 0.87 and 4.5 uM at rat ASIC1a+3, ASIC1a+2a and ASIC2a+3; IC5O values are 0.33 and 0.69 uM at human ASIC1a+2a and ASIC1a+3, with no effect at ASIC2a+3). Attenuates pathophysiological nociceptive behaviors in CFA-inflamed and CCI rats.

Cas No.

309711-59-9

分子式

C19H19N3O2

分子量

321.37

别名

NS 383

储存和溶解度

DMSO:1.61 mg/mL(5 mM)
Powder: -20°C for 3 years
In solvent: -80°C for 2 years