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NRA-0160
本产品不向个人销售,仅用作科学研究,不用于任何人体实验及非科研性质的动物实验。
NRA-0160图片
CAS NO:204718-47-8
包装:5 mg
市场价:7000元

产品介绍

产品描述

NRA-0160 is a selective antagonist of dopamine D4 receptor(Ki of 0.48 nM)

体内活性

NRA0160 dose-dependently and significantly reverses the effects of MAP on both A9 and Al0 dopamine neurons.?NRA0160 is slightly more potent in reversiig the effects of MAP on A10 (ED50 = 1.0 mg/kg) than on A9 dopamine neurons (ED50 = 1.3 mg/kg).?NRA0160 reverses the effect of AP0 on both A9 and A10 dopamine neurons.?ED50 values for the effects of NRA0160 on APO-induced inhibition of A9 and A10 dopamine neurons are 1.3 mg/kg and 0.5 mg/kg, respectively[2].

Cas No.

204718-47-8

分子式

C24H23F2N3OS

分子量

439.52

别名

NRA-0160

储存和溶解度

(< 1 mg/ml refers to the product slightly soluble or insoluble )
Powder: -20°C for 3 years
In solvent: -80°C for 2 years