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Clocapramine
本产品不向个人销售,仅用作科学研究,不用于任何人体实验及非科研性质的动物实验。
Clocapramine图片
CAS NO:47739-98-0
包装:5 mg
市场价:10227元

产品名称
3-Chlorocarpipramine
Clocarpramine
产品介绍

产品描述

Clocapramine is a D2 and 5-HT2A receptors antagonist.

体外活性

In vitro, Clocapramine shows a higher affinity for 5-HT2A than for D2-receptors and has a moderate affinity for D2-receptors.

体内活性

Clocapramine shows the lowest potency for D2-occupancy in vivo [1]. Clocapramine produces ratios of potency in occupying 5-HT2 versus D2 receptors that fall between these two groups (ED50: 14.5 mg/kg for D2, 4.9 mg/kg for 5-HT2) [2].

Cas No.

47739-98-0

分子式

C28H37ClN4O

分子量

481.07

别名

3-Chlorocarpipramine;Clocarpramine;Clocapramine

储存和溶解度

(< 1 mg/ml refers to the product slightly soluble or insoluble )
Powder: -20°C for 3 years
In solvent: -80°C for 2 years