JP1302 dihydrochloride 是一种选择性的、高亲和力的α2C肾上腺受体拮抗剂,其 Kb=16 nM,Ki=28 nM。
产品描述
JP1302 dihydrochloride is a selective, high affinity antagonist of the alpha2C-adrenoceptor (α2C-adrenoceptor), with a Ki (binding affinity) value of 28 nM and a Kb value (antagonist activity) of 16 nM.
Cas No.
1259314-65-2
分子式
C24H26Cl2N4
分子量
441.4
别名
JP1302 dihydrochloride
储存和溶解度
H2O:12 mg/mL (27.18 mM),Need ultrasonic
DMSO:5 mg/mL (11.33 mM),ultrasonic and adjust pH to 5 with NaOH
Powder: -20°C for 3 years
In solvent: -80°C for 2 years