SB271046 是一种强效、选择性和口服活性的 5-HT6 受体拮抗剂,pKi 为 8.9,比其他 5-HT 受体亚型选择性高 200 倍。
产品描述
SB271046 is a potent, selective and orally active 5-HT6 receptor antagonist with pKi of 8.9, exhibits 200-fold greater selectivity over other 5-HT receptor subtypes.
Cas No.
209481-20-9
分子式
C20H23Cl2N3O3S2
分子量
488.44
别名
SB271046
储存和溶解度
H2O:<1 mgml
Ethanol:<1 mgml
DMSO:40 mg/mL (88.49 mM)
Powder: -20°C for 3 years
In solvent: -80°C for 2 years