RET-IN-3 (compound 34) 是一种选择性RETV804M激酶抑制剂(IC50 = 19 nM)。
产品描述
RET-IN-3 (compound 34) is a selective RETV804M kinase inhibitor(IC50 = 19 nM) [1].
体外活性
RET-IN-3 shows 16 and 410 fold selectivity compared to wt-RET and KDR, respectively [1].
Cas No.
2414374-53-9
分子式
C18H21N5O2
分子量
339.39
别名
RET-IN-3
储存和溶解度
(< 1 mg/ml refers to the product slightly soluble or insoluble )
Powder: -20°C for 3 years
In solvent: -80°C for 2 years