CAY10761 is an inhibitor of ectonucleotide pyrophosphatase/phosphodiesterase 1 (ENPP1; IC50s = 467 and 429 μM for the human and snake venom enzymes, respectively).1,2 It also inhibits mushroom tyrosinase (Ki = 1.9 μM) and urease from jack bean, P. mirabilis, and B. pasteurii (IC50s = 0.093,<0.125, and 0.089 mM, respectively, at pH 8.2).3,4

333409-31-7

C7H8N4O2S2

244.29

CAY10761;CAY10761

DMF:30 mg/mL
DMSO:30 mg/mL
DMSO:PBS (pH 7.2) (1:4):0.20 mg/mL
Powder: -20°C for 3 years
In solvent: -80°C for 2 years