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Iodophenpropit dihydrobromide
本产品不向个人销售,仅用作科学研究,不用于任何人体实验及非科研性质的动物实验。
Iodophenpropit dihydrobromide图片
CAS NO:145196-87-8
包装:5 mg
市场价:7000元

产品介绍

产品描述

Iodophenpropit dihydrobromide is an effective and selective antagonist of the histamine H3 receptor. The binding of [125I]Iodophenpropit is readily reversible, selective, and of high affinity (KD: 0.32 nM).

体外活性

Iodophenpropit suppresses 5-hydroxytryptamine (5-HT) responses (IC50 of 1.57±0.3 μM)[3]. Iodophenpropit is a very potent H3 receptor antagonist and displays only a moderate affinity for the H1 and H2 receptors [2].

体内活性

In rabbits, Iodophenpropit (1 μg/kg; through intramuscular; b.i.d.; for 10 days) displays obviously enhancement of total anti-sheep red blood cells (SRBC)- immunoglobulins (Igs)[4].

Cas No.

145196-87-8

分子式

C15H20BrIN4S

分子量

495.22

别名

Iodophenpropit dihydrobromide

储存和溶解度

(< 1 mg/ml refers to the product slightly soluble or insoluble )
Powder: -20°C for 3 years
In solvent: -80°C for 2 years