VU 0255035 是高度选择性、竞争性和血脑屏障通透性的毒蕈碱 M1 受体拮抗剂，IC50为 130 nM，可减少毛果芸香碱诱导的小鼠癫痫发作。

VU 0255035 is a highly selective, competitive and brain penetrant muscarinic M1 receptor antagonist with an IC50 of 130 nM. It reduces pilocarpine-induced seizures in mice. It is used to examine the role of the M1 receptor in diverse situations.

1135243-19-4

C18H20N6O3S2

432.52

VU 0255035

DMSO:Soluble
Powder: -20°C for 3 years
In solvent: -80°C for 2 years