ART-IN-1 (compound 7) 是一种PARP的选择性抑制剂,对 PARP2, TNKS2, PARP10, PARP14, PARP15 的IC50值分别为 19, 22, 2.4, >100, 1.1 μM。
产品描述
ART-IN-1 (compound 7) is a selective inhibitor of PARP with IC 50 s of 19, 22, 2.4, >100, 1.1 μM for PARP2, TNKS2, PARP10, PARP14, PARP15, respectively [1].
体外活性
ART-IN-1 (compound 7) (0-100 μM) is an analog of TIQ-A which shows inhibition of PARP2, TNKS2, PARP10, PARP14, PARP15 with IC 50 s of 19, 22, 2.4, >100, 1.1 μM, respectively [1].
Cas No.
2418014-98-7
分子式
C14H13NO2S
分子量
259.32
储存和溶解度
(< 1 mg/ml refers to the product slightly soluble or insoluble )
Powder: -20°C for 3 years
In solvent: -80°C for 2 years