CAY10727 is an inhibitor of protein arginine deiminase 3 (PAD3; kinact/KI= 15,600 M-1min-1).1It is selective for PAD3 over PAD1, -2, and -4 (kinact/KIs = 360, 1,110, and 1,460 M-1min-1, respectively).

1671088-84-8

C21H22Cl2N4O2

433.33

DMSO:30 mg/mL
DMSO:PBS (pH 7.2) (1:1):0.5 mg/mL
Ethanol:10 mg/mL
DMF:30 mg/mL
Powder: -20°C for 3 years
In solvent: -80°C for 2 years