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(-)-MK 801 Maleate
本产品不向个人销售,仅用作科学研究,不用于任何人体实验及非科研性质的动物实验。
(-)-MK 801 Maleate图片
CAS NO:121917-57-5
包装与价格:
包装价格(元)
25mg电议
50mg电议
100mg电议

产品名称
MK801, MK-801
产品介绍

生物活性

(-)-MK 801 maleate是一种有效的、选择性的、非竞争性的NMDA受体拮抗剂。它通过与NMDA相关离子通道内的一个位点结合而起作用。

靶点信息

NMDA Receptor
30.5 nM(Ki)

化学数据

目录号A13435
作用机制Antagonist (拮抗剂)
M. Wt337.37
FormulaC16H15NC4H4O4
Purity>99%
Storage

Store lyophilized at -20ºC, keep desiccated.
In lyophilized form, the chemical is stable for36 months.
In solution, store at -20ºC and use within3 monthsto prevent loss of potency. Aliquot to avoid multiple freeze/thaw cycles.

CAS No.121917-57-5
SynonymsMK801, MK-801
SMILESC[C@]12C3=CC=CC=C3C[C@H](N1)C4=CC=CC=C24.C(=C/C(=O)O)\C(=O)O

溶解度

In vitro (25°C)DMSO63 mg/mL (186.73 mM)
WaterInsoluble
Ethanol7 mg/mL (20.74 mM)
In vivo2% DMSO+40% PEG 300+2% Tween 80+ddH2O7 mg/mL
*<1 mg/ml means slightly soluble or insoluble.
*Please note that Adooq tests the solubility of all compounds in-house, and the actual solubility may differ slightly from published values. This is normal and is due to slight batch-to-batch variations.

储备液配制

Concentration / Solvent Volume / Mass1 mg5 mg10 mg
0.1 mM29.64 mL148.21 mL296.41 mL
0.5 mM5.93 mL29.64 mL59.28 mL
1 mM2.96 mL14.82 mL29.64 mL
5 mM0.59 mL2.96 mL5.93 mL

*The above data is based on the productmolecular weight 337.37. Batch specific molecular weights may vary from batch to batch due to solvent of hydration, which will affect the solvent volumes required to prepare stock solutions.