CDK7/12-IN-1 是一种选择性CDK7/12抑制剂，对 CDK7 和 CDK 12 的IC50分别为 3 和 277 nM。抑制 CDK7 和 CDK12 是抑制肿瘤生长的有效策略。

CDK7/12-IN-1 is a selective CDK7/12 inhibitor with IC 50 s of 3 and 277 nM for CDK7 and CDK 12, respectively. CDK7 and CDK12 inhibition is an effective strategy to inhibit tumour growth [1].

2654075-94-0

C25H34N8O

462.59

(< 1 mg/ml refers to the product slightly soluble or insoluble )
Powder: -20°C for 3 years
In solvent: -80°C for 2 years