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QCA570
本产品不向个人销售,仅用作科学研究,不用于任何人体实验及非科研性质的动物实验。
QCA570图片
CAS NO:2207569-08-0
包装与价格:
包装价格(元)
5 mg电议
10 mg电议

产品介绍

产品描述

QCA570 is an effective BET degrader based on PROTAC (IC50: 10 nM for BRD4 BD1 Protein).

体外活性

QCA570 inhibits cell growth in MV4;11, MOLM-13, and RS4;11 cell lines (IC50: 8.3, 62, and 32 pM, respectively). QCA570 is an extremely effective and highly efficacious BET degrader, capable of degrading BET proteins at low picomolar (pM) concentrations in leukemia cells. [1].

Cas No.

2207569-08-0

分子式

C39H33N7O4S

分子量

695.79

储存和溶解度

(< 1 mg/ml refers to the product slightly soluble or insoluble )
Powder: -20°C for 3 years
In solvent: -80°C for 2 years