PROTAC BET degrader-2 is a highly potent degrader of Bromodomain and Extra-Terminal (BET) proteins (IC50 of 9.6 nM ).

PROTAC BET degrader-2 is a highly potent Bromodomain and Extra-Terminal (BET) proteins degrader (IC50 value of 9.6 nM in cell growth inhibition in the RS4);11 cells and capable of achieving tumor regression[1].

2093388-33-9

C41H42N10O6

770.84

DMSO:50 mg/mL (64.86 mM),Need ultrasonic
Powder: -20°C for 3 years
In solvent: -80°C for 2 years