A-205804 是一种选择性口服有效的先导抑制剂，抑制E-selectin和ICAM-1表达，IC50分别为 20 nM 和 25 nM，可用于慢性炎症疾病的研究。

A-205804 is a specific and effective inhibitor of E-selectin( IC50=20 nM ) and ICAM-1(IC50=25 nM) expression.

在人内皮细胞中,A-205804选择性抑制ICAM-1(IC50 = 10 nM)和E-selectin (IC50 = 20 nM)。

251992-66-2

C15H12N2OS2

300.41

Ethanol:3 mg/mL (10 mM)
DMSO:30 mg/mL (100 mM)
Powder: -20°C for 3 years
In solvent: -80°C for 2 years