BCTC是有效的、特异性的瞬时受体阳离子通道M8(TRPM8)抑制剂。

BCTC is a potent TRPV1 antagonist that inhibits capsaicin-induced and acid-induced activation of rat TRPV1 (IC50 of 35 and 6 nM, respectively)

393514-24-4

C20H25ClN4O

372.89

N-(4-叔丁苯基)-4-(3-氯吡啶-2-基)哌嗪-1-甲酰胺

DMSO:50 mg/mL (134.09 mM)
Powder: -20°C for 3 years
In solvent: -80°C for 2 years