PF-02575799 is an inhibitor of microsomal triglyceride transfer protein (MTP) (IC50: 0.77±0.29 nM).

PF-02575799 obviously enhance alanine transaminase at 100 mg/kg. PF-02575799 produces appreciable triglyceride effects at its minimally effective dose (10 mg/kg) .

863491-70-7

C42H37FN4O4

680.77

(< 1 mg/ml refers to the product slightly soluble or insoluble )
Powder: -20°C for 3 years
In solvent: -80°C for 2 years