MRS 1754 是A2B腺苷受体选择性拮抗剂，对人和大鼠的 A1和 A3受体的亲和力非常低。

MRS 1754 is a selective antagonist radioligand for the A2B adenosine receptor. It has a very low affinity for A1 and A3 receptors of both humans and rats.

The Ki value for displacement of [3H]MRS 1754 binding to human A2B receptors expressed in HEK-293 cell membranes is 1.45±0.21 nM. The most effective displacer of [3H]MRS 1754 binding is MRS 1754. .

264622-58-4

C26H26N6O4

486.52

DMSO:15 mg/mL (30.83 mM),Need ultrasonic
Powder: -20°C for 3 years
In solvent: -80°C for 2 years