A2A receptor antagonist 1是腺苷A2A和A1受体的拮抗剂，Ki值分别为4和264 nM。

A2A receptor antagonist 1 is an antagonist of both adenosine A2A receptor and A1 receptor with Kis of 4 and 264 nM, respectively.

A2A receptor anyagonist 1 is a potent adenosine A2A receptor antagonist, selective over the A1 receptor and demonstrate its binding activity with Ki values of 4 and 264 nM, respectively. [1]

443103-97-7

C16H12FN5O

309.3

CPI-444 analog;A2A receptor antagonist 1

DMSO:62 mg/mL (200.45 mM)
Powder: -20°C for 3 years
In solvent: -80°C for 2 years