MRS-1706 是一种选择性A2B腺苷受体的反向激动剂，对人 A2B、A2A、A1和 A3受体的Ki值分别为 1.39、112、157 和 230 nM。

MRS-1706 has Ki values of 1.39, 112, 157, and 230 nM for human A2B, A2A, A1, and A3 receptors respectively. MRS-1706 is an effective and selective adenosine A2B receptor inverse agonist.

264622-53-9

C27H29N5O5

503.55

DMSO:6.4 mg/mL (12.71 mM),Need ultrasonic and warming
H2O:< 0.1 mg/mL (insoluble)
Powder: -20°C for 3 years
In solvent: -80°C for 2 years