CaMKII-IN-1是高效的CaMKII选择性抑制剂，IC50为63nM，对CaMKIV, MLCK, p38a, Akt1,和PKC这些靶点几乎无作用。

CaMKII-IN-1 is a potent and highly selective inhibitor of CaMKII (IC50 = 63 nM). CaMKII-IN-1 exhibited more than 100-fold higher selectivity for CaMKII over CaMKIV, MLCK, p38a, Akt1, and PKC.

1208123-85-6

C29H30ClN5O2S

548.1

DMSO:54 mg/mL (98.52 mM)
Powder: -20°C for 3 years
In solvent: -80°C for 2 years