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AR-M 1000390 hydrochloride
本产品不向个人销售,仅用作科学研究,不用于任何人体实验及非科研性质的动物实验。
AR-M 1000390 hydrochloride图片
CAS NO:209808-47-9
包装与价格:
包装价格(元)
2 mg电议
5 mg电议
10 mg电议
50 mg电议
100 mg电议
1 mL*10 mM(in DMSO)电议

产品名称
ARM390 Hydrochloride
ARM-390 HCl
产品介绍
AR-M 1000390 hydrochloride 是选择性 δ 阿片受体激动剂,EC50为 7.2±0.9 nM。

产品描述

AR-M 1000390 (hydrochloride), also known as ARM-390, is a low-internalizing nonpeptidic δ-selective opioid receptor agonist; derivative of SNC 80. Does not trigger acute desensitization of the analgesic response; reduces CFA-induced hyperalgesia. Brain penetrant following systemic administration.

体外活性

Does not trigger acute desensitization of the analgesic response

体内活性

Reduces CFA-induced hyperalgesia. Brain penetrant following systemic administration.

Cas No.

209808-47-9

分子式

C23H29ClN2O

分子量

384.95

别名

ARM390 Hydrochloride;ARM-390 HCl

储存和溶解度

H2O:38.49 mg/mL (100 mM)
DMSO:38.49 mg/mL (100 mM)
Powder: -20°C for 3 years
In solvent: -80°C for 2 years