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Brofaromine
本产品不向个人销售,仅用作科学研究,不用于任何人体实验及非科研性质的动物实验。
Brofaromine图片
CAS NO:63638-91-5
包装与价格:
包装价格(元)
50 mg电议
100 mg电议

产品名称
CGP 11305A
产品介绍

产品描述

Brofaromine (CGP 11305A) is an MAO inhibitor (IC50: 0.2 μM for MAO-A).

体外活性

In order to assess whether the protective effect is related to the inhibition of the MAO-A or due to another mechanism, the effect of Brofaromine is determined on the activity of MAO-A in cultured cortical cells. The cultured cortical cells have significant MAO-A activity. Brofaromine inhibits the enzyme in a concentration-dependent manner (IC50: 0.19?μM). Hill coefficient is 0.96. The enzyme is almost completely inhibited at 10?μM. Brofaromine inhibits MAO-A activity of our cultured cortical cells in a concentration-dependent manner. The IC50 range of Brofaromine is 0.01?μM to 0.1?μM.

Cas No.

63638-91-5

分子式

C14H16BrNO2

分子量

310.19

别名

CGP 11305A

储存和溶解度

DMSO:250 mg/mL (805.96 mM),Need ultrasonic
Powder: -20°C for 3 years
In solvent: -80°C for 2 years