Ocinaplon 是一种GABAA受体的阳性变构调节剂,在 α1 亚基处有较高的活性。
产品描述
Ocinaplon is a GABAA receptors modulator.
体内活性
In rats, ocinaplon produces significant muscle relaxation, ataxia, and sedation only at doses >25-fold higher than the minimum effective dose (3.1 mg/kg) in the Vogel "conflict" test[2].
Cas No.
96604-21-6
分子式
C17H11N5O
分子量
301.3
别名
奥西普隆;DOV 273547
储存和溶解度
DMSO:<1 mgml
2eq.HCl:<25mg>Powder: -20°C for 3 years
In solvent: -80°C for 2 years