CGP52432 是一种GABAB受体拮抗剂,IC50值为 85 nM。
产品描述
CGP52432 is a very potent antagonist of GABAB receptors (IC50 = 85 nM).
激酶实验
Reactions are set up with Acetyl coenzyme A (AcCoA)(0.4 μM), N-terminal histone H4 peptide (sequence SGRGKGGKGLGKGGAKRHRKV-GGK-biotin)(50 nM), MOZ enzyme(10 nM), and an acetyl-lysine specific antibody (final dilution 1: 10000).
Cas No.
139667-74-6
分子式
C15H24Cl2NO4P
分子量
384.23
别名
CGP 52432;4-苄氧基苯基异硫氰酸酯
储存和溶解度
DMSO:5 mg/mL (13.01 mM),Need ultrasonic and warming
Powder: -20°C for 3 years
In solvent: -80°C for 2 years