Vofopitant dihydrochloride is a selective and orally available antagonist of tachykinin neurokinin 1(NK1) receptor (pKi: 9.5 and 10.6 in rat and human membranes respectively) and is a potential broad-spectrum anti-emetic agent.

168266-51-1

C21H25Cl2F3N6O

505.36

GR 205171A

(< 1 mg/ml refers to the product slightly soluble or insoluble )
Powder: -20°C for 3 years
In solvent: -80°C for 2 years