Scyliorhinin II acetate 是大鼠大脑皮层神经激肽 3 (NK3) 受体 (Ki = 2.5 nM) 的选择性激动剂。
产品描述
Scyliorhinin II acetate is a selective agonist of the neurokinin-3 (NK3) receptor (Ki = 2.5 nM) in rat cerebral cortex.
体外活性
Scyliorhinin II acetate has little effect on NK1 and NK2 receptors. The Ki values for NK1/NK3 and NK2/NK3 are 176 and 200, respectively[2].
体内活性
In mice, Scyliorhinin II acetate(i.c.v.) produced potent and dose-related reciprocal hindlimb scratching about equipotently (ED50 = 0.08 nmol)[1].
Cas No.
TP1851L
储存和溶解度
(< 1 mg/ml refers to the product slightly soluble or insoluble )
Powder: -20°C for 3 years
In solvent: -80°C for 2 years