Trimipramine maleate 是一种 5-HT 受体拮抗剂，对 5-HT1C、5-HT2和 5-HT1A受体的 pKi值分别为 6.39、8.10和 4.66。

Trimipramine maleate appears to inhibit serotonin transport and norepinephrine uptake by nerve terminals. This increases available norepinephrine or serotonin and prolongs its action. Trimipramine Maleate is the maleate salt form of trimipramine, a tricyclic secondary amine of the dibenzazepine class, with an antidepressant property.

521-78-8

C24H30N2O4

410.514

Surmontil maleate;马来酸三甲丙咪嗪;三甲丙咪嗪马来酸盐

DMSO:10 mM
Powder: -20°C for 3 years
In solvent: -80°C for 2 years