Jaspamycin (7-CN-7-C-Ino) does not bind with purified human PKARIα. Anti-parasite activity. Jaspamycin (7-CN-7-C-Ino) is a potent activator of PKA, binding to the R site (PKAR), with an EC50 of 6.5 nM and Kd of 8 nM in Trypanosoma brucei.

22242-96-2

C12H12N4O5

292.25

7-CN-7-C-Ino

DMSO:41.67 mg/mL (142.58 mM),Need ultrasonic
Powder: -20°C for 3 years
In solvent: -80°C for 2 years