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VBY-825
本产品不向个人销售,仅用作科学研究,不用于任何人体实验及非科研性质的动物实验。
VBY-825图片
CAS NO:1310340-58-9
包装与价格:
包装价格(元)
1 mg电议
2 mg电议
5 mg电议
10 mg电议
100 mg电议

产品介绍
VBY-825是CAThepsin一种新型的可逆抑制剂,对CAThepsin B, L, S和V都有很高的抑制力。

产品描述

VBY-825 is a reversible inhibitor of cathepsin with high potency against cathepsins B, L, S and V.

体外活性

VBY-825 is a potent assayed cathepsins inhibitor and its potency against at least one cathepsin, cathepsin S, extends across species relevant for pharmacology studies, specifically mouse. 10 mg/kg/day dose of VBY-825 achieves a trough plasma concentration >200nM, which is well above that required for full inhibition of the intracellular activity of cathepsins B, F, K, L, S and V in both mouse and human cell lines.

Cas No.

1310340-58-9

分子式

C23H29F4N3O5S

分子量

535.55

储存和溶解度

DMSO:125 mg/mL (233.40 mM),Need ultrasonic
Powder: -20°C for 3 years
In solvent: -80°C for 2 years