ObafiSTAT 是醛酮还原酶AKR1C3的有效抑制剂,抑制人 AKR1C3 的IC50为 1.2 nM。
产品描述
Obafistat is a potent inhibitor of aldo-keto reductase AKR1C3 with an IC50 of 1.2 nM for human AKR1C3 (patent WO2017202817A1, example 4).
Cas No.
2160582-57-8
分子式
C15H16FN5O3S
分子量
365.38
储存和溶解度
DMSO:62.5 mg/mL (171.05 mM),Need ultrasonic and warming and heat to 60°C
Powder: -20°C for 3 years
In solvent: -80°C for 2 years